- Chemo-enzymatic synthesis of ester-linked docetaxel-monosaccharide conjugates as water-soluble prodrugs
-
Three new docetaxel prodrugs, i.e., 7-propionyldocetaxel 3′′-O-β-D-glycopyranosides, which contain ester-linked monosaccharides, were synthesized by a chemo-enzymatic procedure involving enzymatic transglycosylations with lactase, b-galactosidase, or β-xy
- Shimoda, Kei,Kubota, Naoji
-
p. 6769 - 6777
(2011/11/07)
-