Mechanistic Duality of Bacterial Efflux Substrates and Inhibitors: Example of Simple Substituted Cinnamoyl and Naphthyl Amides
Antibiotic resistance poses an immediate and growing threat to human health. Multidrug efflux pumps are promising targets for overcoming antibiotic resistance with small-molecule therapeutics. Previously, we identified a diaminoquinoline acrylamide, NSC-3
Cao, Feng,Cooper, Connor J.,D'Cunha, Napoleon,Haynes, Keith,Leus, Inga V.,Malloci, Giuliano,Margiotta, Enrico,Moniruzzaman, Mohammad,Parks, Jerry M.,Ruggerone, Paolo,Rybenkov, Valentin V.,Uddin, Muhammad R.,Vargiu, Attilio V.,Walker, John K.,Zgurskaya, Helen I.