Studies on the Claisen rearrangements in the indolo[2,3-b]quinoline system
A study of the effect of substrate structure on a Claisen-aza-Cope reaction is presented including a rationalisation of the reaction outcome using DFT calculations. An asymmetric version of the reaction is also described that is of relevance to a proposed
Voute, Nicholas,Philp, Douglas,Slawin, Alexandra M. Z.,Westwood, Nicholas J.
supporting information; experimental part
p. 442 - 450
(2010/02/16)
Drug design, in vitro pharmacology, and structure-activity relationships of 3-acylamino-2-aminopropionic acid derivatives, a novel class of partial agonists at the glycine site on the N-methyl-D-aspartate (NMDA) receptor complex
Retaining agonistic activity at the glycine coagonist site of the NMDA receptor in molecules derived from glycine or D-serine has proven to be difficult because in the vicinity of the α-amino acid group little substitution is tolerated. We have solved thi
Urwyler, Stephan,Floersheim, Philipp,Roy, Bernard L.,Koller, Manuel
supporting information; experimental part
p. 5093 - 5107
(2010/03/02)
A CONVENIENT SYNTHETIC APPROACH TO 4-SUBSTITUTED INDOLES
A simple and practical synthetic method for 4-halogenoindoles, 4-indolecarbaldehyde, 4-cyanoindole, and 4-methoxycarbonylindole is elaborated.
Yamada, Fumio,Somei, Masanori
p. 1173 - 1176
(2007/10/02)
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