- BENZOXAZINONE AND BENZOXAZEPINONE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS
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The present invention provides a compound of formula (I) wherein X is a structure of the following formula (i), (ii), (iii), or iv G is O, or S; U is -(CR3R4)n-; W is CH2NHC(=G)R1, CH2NH-het, CH2-G-het, CH2het, C(=O)NHR2; and Y1, Y2 and Y3 are independently CH, or CF. The compounds of the present invention are useful as antibacterial agents.
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(2010/11/28)
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- 2,2-dimethyl-3-(but-1-en-3-ynyl)-cyclopropane carboxylates
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Compounds of the formula STR1 wherein X is hydrogen, halogen or an optionally substituted alkyl, Y is selected from the group consisting of hydrogen, halogen optionally substituted alkyl, an optionally substituted aryl or arylalkyl, --(CH2)sub
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- Esters of 2,2-dimethyl-3-[(2,2-difluoro-cyclopropylidene) methyl]cyclopropane carboxylic acids
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A compound selected from the group consisting of all stereoisomeric forms and mixtures thereof of a compound of the formula STR1 wherein Y and Z are individually selected from the groups consisting of hydrogen, halogen, --CF3, alkyl, alkoxy and alkylthio of 1 to 8 carbon atoms and aryl, aryloxy and arylthio of up to 14 carbon atoms optionally substituted with at least one member of the group consisting of halogen, hydroxy optionally esterified etherified, --CF3 and alkyl of 1 to 8 carbon atoms and R is alkyl of 1 to 8 carbon atoms or the remainder of a pyrethrinoid alcohol having excellent pesticidal properties and their preparation and intermediates.
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- 1-cyclopropyl-6-fluoro-8-alkyl-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives
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Novel 4-oxoquinoline-3-carboxylic acid compounds of the formula: STR1 wherein R2 is 1-pyrrolidinyl which may have 1 to 2 substituents selected from the group consisting of (i) C1 -C6 alkyl, (ii) amino-(C1 -Csub
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- 1-Cyclopropyl-6-fluoro-7-piperazinyl-1,4-Dihydro-4-oxo-quinoline-3-carboxylic acid derivatives
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Novel 4-oxoquinoline-3-carboxylic acid compounds of the formula: STR1 wherein R2 is a heterocyclic group: STR2 in which RA is H, C1 -C6 alkyl or phenyl (C1 -C6) alkyl, RB is 2-ox
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- Benzoheterocyclic compounds
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Novel 4-oxoquinoline-3-carboxylic acid compounds of the formula: STR1 wherein R3 is C1 -C6 alkyl and RF is C1 -C6 alkyl, and a pharmaceutically acceptable salts thereof, said compounds havi
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