- 5- OR 7-AZAINDAZOLES AS BETA-LACTAMASE INHIBITORS
-
The present invention relates to β-lactamase inhibitors having the following general formula (I): wherein R1-R4 and X1-X2 are defined in the specification, pharmaceutical composition thereof, and use thereof for the treatment of a bacterial infection, alone or in combination with β-lactam antibiotics and/or other antibiotics and/or other β-lactamase inhibitors.
- -
-
Page/Page column 41; 43; 44
(2020/09/19)
-
- INHIBITORS OF FATTY ACID BINDING PROTEIN (FABP)
-
The present invention relates to novel heterocyclic compounds as Fatty Acid Binding Protein ("FABP") inhibitors, pharmaceutical compositions comprising the heterocyclic compounds and the use of the compounds for treating or preventing a cardiovascular disease, a metabolic disorder, obesity or an obesity-related disorder, diabetes, dyslipidemia, a diabetic complication, impaired glucose tolerance or impaired fasting glucose. An illustrative compound of the present invention is shown below: (I)
- -
-
Page/Page column 159
(2010/06/15)
-
