- THIAZOLE DERIVATIVE AND APPLICATIONS THEREOF
-
Disclosed in the present invention are a new thiazole compound, particularly a compound represented by formula (I), a pharmaceutical composition thereof and applications thereof in the preparation of drugs for the treatment of diseases related to herpes simplex viruses.
- -
-
Paragraph 0096; 0100
(2020/01/02)
-
- Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action
-
A series of congeners structurally related to pritelivir, N-[5-(aminosulfonyl)-4-methyl-1,3-thiazol-2-yl]-N-methyl-2-[4-(2-pyridinyl)phenyl]acetamide, a helicase-primase inhibitor for the treatment of herpes simplex virus infections, was prepared. The syn
- Carta, Fabrizio,Birkmann, Alexander,Pfaff, Tamara,Buschmann, Helmut,Schwab, Wilfried,Zimmermann, Holger,Maresca, Alfonso,Supuran, Claudiu T.
-
p. 3154 - 3164
(2017/04/19)
-
- APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
-
Disclosed are compounds which inhibit the activity of anti-apoptotic Bcl-2 proteins, compositions containing the compounds and methods of treating diseases during which is expressed anti-apoptotic Bcl-2 protein.
- -
-
Page/Page column 56
(2010/08/07)
-
- Acetylenyl-pyrazolo-pyrimidine derivatives
-
The present invention relates to compounds of formula (I): wherein R1 to R3, A, M, L, E, G, and J are as defined in the description and claims. The invention also relates to a process for the manufacture of such compounds, pharmaceutical compositions containing them, and methods for treating CNS disorders.
- -
-
Page/Page column 29
(2008/06/13)
-
- Thiazolyl amide derivatives
-
The present invention relates to novel compounds, to a process for their preparation and to their use as medicaments, in particular as antiviral medicaments.
- -
-
-
- Inverse thiazolylamide derivatives
-
The present invention relates to novel compounds, i.e. inverse thiazolylamide derivatives, to processes for their preparation and to their use as medicaments, in particular as antiviral medicaments.
- -
-
-