- MOSQUITO VECTOR CONTROL COMPOSITIONS, METHODS AND PRODUCTS UTILIZING SAME
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The present inventions concerns use of a certain methoxyacrylate compound to control mosquitoes, and vector control solutions comprising a defined methoxyacrylate compound, in particular the invention relates to a substrate, to a composition, for controll
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Page/Page column 39
(2016/12/22)
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- CARBACEPHEM β-LACTAM ANTIBIOTICS
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Carbacephem -lactam antibiotics having structure (I) are disclosed, including stereoisomers, pharmaceutically acceptable salts, esters and prodrugs thereof, wherein Ar1, Ar2, R1 and R2 are as defined herein. The compounds are useful for the treatment of bacterial infections, in particular those caused by methicillin-resistant Staphylococcus spp.
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Page/Page column 90
(2010/04/06)
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- CARBACEPHEM BETA-LACTAM ANTIBIOTICS
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Carbacephem β-lactam antibiotics having chemical structures (I) and (II) are disclosed: including stereoisomers, pharmaceutically acceptable salts, esters and prodrugs thereof, wherein Ar2, R1, R2 and R6 are as defined herein. The compounds are useful for the treatment of bacterial infections, in particular those caused by methicillin-resistant Staphylococcus spp.
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Page/Page column 64
(2010/11/05)
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- Novel, potent P2-P3 pyrrolidine derivatives of ketoamide-based cathepsin K inhibitors
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Starting from a potent pantolactone ketoamide cathepsin K inhibitor discovered from structural screening, conversion of the lactone scaffold to a pyrrolidine scaffold allowed exploration of the S3 subsite of cathepsin K. Manipulation of P3
- Barrett, David G.,Catalano, John G.,Deaton, David N.,Hassell, Anne M.,Long, Stacey T.,Miller, Aaron B.,Miller, Larry R.,Ray, John A.,Samano, Vicente,Shewchuk, Lisa M.,Wells-Knecht, Kevin J.,Willard Jr., Derril H.,Wright, Lois L.
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p. 1735 - 1739
(2007/10/03)
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- 2-Substituted-5-trifluoromethyl-1,3,4-thiadiazoles
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2-Substituted-5-trifluoromethyl-1,3,4-thiadiazoles of the formula STR1 in which R is substituted alkyl, phenyl monosubstituted in the o- or m- position, polysubstituted phenyl, substituted phenylalkyl, phenylalkenyl, substituted phenylalkenyl, an optionally substituted 5-membered or 6-membered heterocyclic radical with 1 to 4 hetero-atoms selected from N and S atoms, optionally substituted benzimidazolyl or benzthiazolyl, optionally substituted naphthyl, quinolyl, cyano or one of the groups STR2 wherein R1 and R2 conjointly are a trimethylene, tetramethylene or pentamethylene group, X is oxygen or sulfur, R' and R" each independently is alkyl or, together with the nitrogen atom and optionally further hetero-atoms selected from O and N atoms, form an optionally substituted 6-membered or 7-membered ring, and N is 0, 1 or 2, Which possess fungicidal, bactericidal, arthropodicidal and insecticidal properties.
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