Use of a modified Leimgruber-Batcho reaction to prepare 6-chloro-5-fluoroindole
An efficient synthesis of the title indole, the heterocyclic core of the standard 5-HT2C receptor agonist Ro 60-0175, via a modified Leimgruber-Batcho indole synthesis is presented. The process can be used to make > 100 g quantities of the targ
Bentley, Jon M.,Davidson, James E.,Duncton, Matthew A. J.,Giles, Paul R.,Pratt, Robert M.
p. 2295 - 2300
(2007/10/03)
Stereoselective in vitro aromatic ring oxygenations of chiral 1,4 benzodiazepin 2 ones
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Kolbah,Blazevic,Hannoun,et al.
p. 265 - 283
(2007/10/08)
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