- Solid-phase synthesis of 1,3-azole-based peptides and peptidomimetics
-
We report highly efficient two-step procedures for the synthesis of 1,3-oxazole-, thiazole-, and imidazole-containing peptides on solid phase from dipeptides composed of C-terminal threonine, serine, cysteine, or diaminopropionic acid by using different cyclodehydration procedures followed or preceded by oxidation. The methods are compatible with Fmoc solid-phase peptide synthesis conditions and with N-Fmoc, N-Boc, N-Cbz, and N-Alloc protecting groups.
- Biron, Eric,Chatterjee, Jayanta,Kessler, Horst
-
p. 2417 - 2420
(2007/10/03)
-
- Chemo-enzymatic synthesis of Fmoc-peptide fragments
-
Optically pure Fmoc-peptide fragments have been prepared via dicyclohexylcarbodiimide coupling of N-protected amino acids with amino cid esters, followed by enzyme-catalyzed ester hydrolysis by alcalase with a high concentration of organic solvent in a hi
- Chen,Hsiao,Chang,Wang
-
p. 391 - 398
(2007/10/02)
-
- Synthesis of 2>- and 6>-Locust Adipokinetic Hormone
-
The syntheses of 2>- and 6>-locust adipokinetic hormone (LAKH) by the coupling of N-terminal hexapeptides prepared by the solid-phase method with a common C-terminal tetrapeptide synthesised in solution
- Hardy, Paul M.,Sheppard, Paul W.
-
p. 723 - 729
(2007/10/02)
-