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R2
R1
O
R3
hydroamination
N
Ar
X
(π*+σ*)
R1
O
electrophore
29 examples
N
weak bond
O
R
transition
metalꢀfree
aryloxyamides
ꢀ easyꢀtoꢀmake
R1 = alkyl, Boc, Cbz
ꢀ
Ar
Nꢀarylation
R1
N
O
R
22 examples
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