Journal of Medicinal Chemistry p. 4964 - 4975 (2015)
Update date:2022-08-15
Topics:
Vincetti, Paolo
Caporuscio, Fabiana
Kaptein, Suzanne
Gioiello, Antimo
Mancino, Valentina
Suzuki, Youichi
Yamamoto, Naoki
Crespan, Emmanuele
Lossani, Andrea
Maga, Giovanni
Rastelli, Giulio
Castagnolo, Daniele
Neyts, Johan
Leyssen, Pieter
Costantino, Gabriele
Radi, Marco
This study describes the discovery of novel dengue virus inhibitors targeting both a crucial viral protein-protein interaction and an essential host cell factor as a strategy to reduce the emergence of drug resistance. Starting from known c-Src inhibitors
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