Journal of Medicinal Chemistry p. 2079 - 2084 (1994)
Update date:2022-08-02
Topics:
Tawada, Hiroyuki
Harcourt, Myles
Kawamura, Noriaki
Kajino, Masahiro
Ishikawa, Eiichiro
et al.
A series of 3-quinolylurea derivatives (1) was synthesized and evaluated for acyl-CoA:cholesterol acyltransferase (ACAT) inhibitory activity.For in vitro studies, the most potent inhibitory activity was found in derivatives having substituents at the 6,7-
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