Journal of Medicinal Chemistry p. 877 - 885 (1992)
Update date:2022-08-04
Topics:
Thomas
Allott
Gibson
Major
Masek
Oldham
Ratcliffe
Roberts
Russell
Thomason
On the basis of an extension of the literature lead 1, a series of benzimidazoles have been synthesized and shown to be angiotensin II (AII) receptor antagonists. The structure-activity relationships of these new antagonists have been explored and the key
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