Journal of Medicinal Chemistry p. 2477 - 2483 (1991)
Update date:2022-07-29
Topics: Selectivity Potency Research and Development Pharmacological Activity Therapeutic Potential
Malleron, Jean-Luc
Comte, Marie-Therese
Gueremy, Claude
Peyronel, Jean Francois
Truchon, Alain
et al.
A series of 2-(aminoalkyl)naphth<1,8-cd>isothiazole 1,1-dioxides was synthesized and examined in various receptor binding tests.Most compounds demonstrated high affinity for the 5-HT2 receptor with moderate to high selectivity.A member of this
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