European Journal of Medicinal Chemistry p. 59 - 76 (2019)
Update date:2022-08-15
Topics:
Pati, Maria Laura
Vitale, Paola
Ferorelli, Savina
Iaselli, Mariaclara
Miciaccia, Morena
Boccarelli, Angelina
Di Mauro, Giuseppe Davide
Fortuna, Cosimo G.
Souza Domingos, Thaisa Francielle
Rodrigues Pereira da Silva, Luiz Cláudio
de Pádula, Marcelo
Cabral, Lucio Mendes
Sathler, Plínio Cunha
Vacca, Angelo
Scilimati, Antonio
Perrone, Maria Grazia
A set of novel diarylisoxazoles has been projected using mofezolac (1) as a lead compound to investigate structure-inhibitory activity relationships of new compounds and the cyclooxygenases (COXs) catalytic activity. Mofezolac was chosen because is the mo
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