Tetrahedron Letters p. 1297 - 1300 (1996)
Update date:2022-09-26
Topics:
Taylor, G. Mark
Baker, Stewart J.
Gedney, Andrea
Pearson, David J.
Sibley, Graham E. M.
The Ritter reactions of 3-alkyl-3-hydroxyazetidine or -piperidine derivatives give low yields of the desired products, whereas the 3-alkyl-3-hydroxy-pyrrolidine and 4-alkyl-4-hydroxy-piperidine derivatives react smoothly to give the corresponding acetamides. An alternative route to 3-acylamino-3-alkylpiperidines, which were designed as conformationally-restricted reduced amide dipeptide isosteres, was devised from nipecotic acid vai a Hofmann rearrangement.
View MoreHebei Kangtai Pharmaceutical Co.,Ltd
Contact:+86-0317-3512963
Address:Wugang Road,Mengcun of Cangzhou City,Hebei Province ,China
Beijing Merson Pharmaceutical Co., Ltd
Contact:0086-10-80484934 0086-10-80484574/
Address:2nd Floor , No. 2 Building , No. 14 Houshayu Duan, Jingmi Road ,Shunyi District , Beijing 101318, P.R.China
Lianyungang Ningkang Chemical Co., Ltd
Contact:.+86-518-88588008
Address:http://www.chemnk.com
TAIXING BEST NEW MATERIALS CO., LTD
Contact:0523-87998158;
Address:No.18 Zhonggang Road,Taixing City ,Jiangsu , China
Contact:17316303296
Address:240 Amboy Ave
Doi:10.1016/j.inoche.2016.10.017
(2016)Doi:10.1021/om9600248
(1996)Doi:10.1021/om980850b
(1999)Doi:10.1016/S0040-4020(96)00339-0
(1996)Doi:10.1016/S0022-328X(00)82760-6
(1968)Doi:10.1016/0968-0896(96)00054-5
(1996)