Bioorganic and Medicinal Chemistry Letters p. 1573 - 1576 (1999)
Update date:2022-08-04
Topics:
Wichmann, Juergen
Adam, Geo
Kolczewski, Sabine
Mutel, Vincent
Woltering, Thomas
A series of 5H-thiazolo[3,2-a]pyrimidine derivatives 1 was studied with respect to the inhibition of 1S,3R-ACPD (10μM)-stimulated GTP γ35S binding on rat mGlu2 receptor transfected cell membranes. The influence of substituents at position 6 and
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