Medicinal Chemistry Research p. 149 - 157 (2004)
Update date:2022-07-30
Topics:
Rawson, David J.
Dack, Kevin N.
Dickinson, Roger P.
James, Kim
Long, Clive
Walker, Don
The potency and pharmacokinetic properties of an indole-based series of endothelin antagonists have been optimised using in vitro, in silico and in vivo methods. Compound 8 is oxidised in vivo to the active metabolite 7 and has been highlighted as an oral
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