Journal of Medicinal Chemistry p. 2391 - 2410 (2020)
Update date:2022-08-15
Topics:
K?se, Meryem
Pillaiyar, Thanigaimalai
Namasivayam, Vigneshwaran
De Filippo, Elisabetta
Sylvester, Katharina
Ulven, Trond
Von Kügelgen, Ivar
Müller, Christa E.
The orphan G protein-coupled receptor (GPCR) GPR84 is expressed on immune cells mediating proinflammatory and immunostimulatory effects. In this study, we prepared the fully efficacious, nonbiased GPR84 agonist 6-hexylamino-2,4(1H,3H)-pyrimidinedione (6)
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