Journal of Medicinal Chemistry p. 3611 - 3625 (2015)
Update date:2022-08-03
Topics:
Boyd, Scott
Brookfield, Joanna L.
Critchlow, Susan E.
Cumming, Iain A.
Curtis, Nicola J.
Debreczeni, Judit
Degorce, Sébastien L.
Donald, Craig
Evans, Nicola J.
Groombridge, Sam
Hopcroft, Philip
Jones, Neil P.
Kettle, Jason G.
Lamont, Scott
Lewis, Hilary J.
MacFaull, Philip
McLoughlin, Sheila B.
Rigoreau, Laurent J. M.
Smith, James M.
St-Gallay, Steve
Stock, Julie K.
Turnbull, Andrew P.
Wheatley, Edward R.
Winter, Jon
Wingfield, Jonathan
A weak screening hit with suboptimal physicochemical properties was optimized against PFKFB3 kinase using critical structure-guided insights. The resulting compounds demonstrated high selectivity over related PFKFB isoforms and modulation of the target in
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