Bioorganic and Medicinal Chemistry Letters p. 2589 - 2592 (2001)
Update date:2022-08-03
Topics:
Folkes, Adrian
Roe, Michael B.
Sohal, Sukhjit
Golec, Julian
Faint, Richard
Brooks, Teresa
Charlton, Peter
We have synthesized and evaluated a series of diketopiperazine-based inhibitors of PAI-1. These studies resulted in the identification of 34 which inhibited PAI-1 in vitro with an IC50 = 0.2 μM. The synthesis and SAR of these compounds are desc
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