Bioorganic Chemistry (2019)
Update date:2022-08-03
Topics:
Huang, Jianping
Huang, Jiaxin
Wang, Ning
Wang, Luhong
Li, Lei
Wang, Changyuan
Sun, Xiuli
Li, Yongming
Huang, Guoping
Ma, Xiaodong
A new class of 2(1H)-pyrimidinone derivatives was identified as potential EGFR T790M inhibitors against TKI-resistant NSCLC. These novel compounds inhibited the EGFR T790M kinase activity at concentrations in the range of 85.3 to 519.9 nM. In particular,
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