Journal of Medicinal Chemistry p. 894 - 900 (1984)
Update date:2022-09-26
Topics:
Heeres
Backx
Van Cutsem
A series of novel triazol-3-ones has been synthesized, and their in vitro and in vivo antifungal properties are reported. Traconazole. which displays a pronounced oral activity against vaginal candidosis in rats and against microsporosis in guinea pigs, has been selected for clinical evaluation.
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