European Journal of Medicinal Chemistry p. 129 - 136 (1991)
Update date:2022-08-02
Topics:
Iskander, MN
Andrews, PR
Winkler, DA
Brinkworth, RI
Paola, C Di
et al.
Our previous calculations on the reaction catalysed by GABA-aminotransferase (GABA-T) have been utilized in this work in order to synthesize a series of reversible inhibitors of this enzyme.The synthesized transition-state analogues and their precursors i
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