1272
I. Collins et al. / Bioorg. Med. Chem. 14 (2006) 1255–1273
13–17, 2005; American Chemical Society: Washington,
DC, 2005; MEDI-143.
the preparation of compound 65, Wendy Blakemore for
assistance with X-ray data collection, Marcel Verdonk
for assistance with molecular modelling studies, Brent
Graham for PKA purification, and Amin Mirza and
Meirion Richards for assistance with compound
characterisation.
14. Gong, J.; Woods, K. W.; Li, T.; Fisher, J.; Packard, G.;
Gandhi, V. B.; Claibone, A.; Luo, Y.; Shi, Y.; Liu, X.;
Klinghofer, V.; Bouska, J.; Shoemaker, A.; Oleksijew, A.;
Jarvis, K.; Stoll, V. S.; Hutchins, C.; De Jong, R.;
Oltersdorf, T.; Li, Q.; Rosenberg, S. H.; Giranda, V. L.;
Zhu, G.-D. Abstracts of Papers, 229th National Meeting
of the American Chemical Society, San Diego, CA, March
13–17, 2005; American Chemical Society: Washington,
DC, 2005; MEDI-142.
15. Giranda, V.; Luo, Y.; Li, Q.; Shoemaker, A.; de Jong,
R.; Liu, X.; Han, E.; Woods, K.; Thomas, S.; Rosen-
berg, S. Eur. J. Cancer Suppl. 2004, 8, 76, Abstracts of
the 16th EORTC-NCI-AACR Symposium on Molecular
Targets and Cancer Therapeutics, Geneva, Switzerland,
2004.
Supplementary material
Supplementary data associated with this article can be
found in the online version at doi:10.1016/
j.bmc.2005.09.055.
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