Journal of Medicinal Chemistry p. 1693 - 1715 (2017)
Update date:2022-08-15
Topics:
Vianello, Paola
Sartori, Luca
Amigoni, Federica
Cappa, Anna
Fagá, Giovanni
Fattori, Raimondo
Legnaghi, Elena
Ciossani, Giuseppe
Mattevi, Andrea
Meroni, Giuseppe
Moretti, Loris
Cecatiello, Valentina
Pasqualato, Sebastiano
Romussi, Alessia
Thaler, Florian
Trifiró, Paolo
Villa, Manuela
Botrugno, Oronza A.
Dessanti, Paola
Minucci, Saverio
Vultaggio, Stefania
Zagarrí, Elisa
Varasi, Mario
Mercurio, Ciro
The balance of methylation levels at histone H3 lysine 4 (H3K4) is regulated by KDM1A (LSD1). KDM1A is overexpressed in several tumor types, thus representing an emerging target for the development of novel cancer therapeutics. We have previously describe
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