Journal of Medicinal Chemistry p. 3407 - 3427 (2019)
Update date:2022-08-15
Topics:
Shirai, Fumiyuki
Tsumura, Takeshi
Yashiroda, Yoko
Yuki, Hitomi
Niwa, Hideaki
Sato, Shin
Chikada, Tsubasa
Koda, Yasuko
Washizuka, Kenichi
Yoshimoto, Nobuko
Abe, Masako
Onuki, Tetsuo
Mazaki, Yui
Hirama, Chizuko
Fukami, Takehiro
Watanabe, Hirofumi
Honma, Teruki
Umehara, Takashi
Shirouzu, Mikako
Okue, Masayuki
Kano, Yuko
Watanabe, Takashi
Kitamura, Kouichi
Shitara, Eiki
Muramatsu, Yukiko
Yoshida, Haruka
Mizutani, Anna
Seimiya, Hiroyuki
Yoshida, Minoru
Koyama, Hiroo
The canonical WNT pathway plays an important role in cancer pathogenesis. Inhibition of poly(ADP-ribose) polymerase catalytic activity of the tankyrases (TNKS/TNKS2) has been reported to reduce the Wnt/β-catenin signal by preventing poly ADP-ribosylation-
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