Journal of Medicinal Chemistry p. 10848 - 10866 (2019)
Update date:2022-08-15
Topics: in vivo Agonists Histamine H3 receptor Non-imidazole 4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines High-Affinity Central Nervous System Activity
Wágner, Gábor
Mocking, Tamara A. M.
Arimont, Marta
Provensi, Gustavo
Rani, Barbara
Silva-Marques, Bruna
Latacz, Gniewomir
Da Costa Pereira, Daniel
Karatzidou, Christina
Vischer, Henry F.
Wijtmans, Maikel
Kie?-Kononowicz, Katarzyna
De Esch, Iwan J. P.
Leurs, Rob
Despite the high diversity of histamine H3 receptor (H3R) antagonist/inverse agonist structures, partial or full H3R agonists have typically been imidazole derivatives. An in-house screening campaign intriguingly afforded
View MoreChongqing maohuan Chemicals Co., Ltd
website:http://www.bschem.com
Contact:+86 13996103726
Address:Chongqing Nan'an District Tu Town
Reliable Pharma Technology (Shanghai) Co., Ltd.
Contact:0086-21-67676847-8008
Address:Lane 1500, No.68, Xinfei Road, Songjiang District, Shanghai, 201611, P.R.China.
shanghai Tauto Biotech Co., Ltd
website:http://www.tautobiotech.com/en/index.htm
Contact:+86-21-51320588 ext. 8025
Address:No. 326, Aidisheng Rd , Zhangjiang Hi-tech Park, Shanghai , P.R.CHINA
Contact:+86--29-82745382
Address:Development Area Of Lantian Country,Xi'an Shanxi.China
Shanghai KFSL Pharmaceutical Technology Co.,Ltd.
Contact:+86-21-39971718
Address:859 jiadingchengliu shanghai
Doi:10.1016/j.tet.2010.04.051
(2010)Doi:10.1016/j.saa.2010.04.019
(2010)Doi:10.1002/adsc.202100112
(2021)Doi:10.1134/S1070428010050234
(2010)Doi:10.1021/om100415z
(2010)Doi:10.1021/ja00206a059
(1989)