Acknowledgments
This work was supported by the National Natural Science
Foundation of China (No. 81172919, 81130023, 31373382),
National Basic Research Plan (973) of the Ministry of Science
and Technology of China (2011CB5C4403), the State Key
Laboratory of Drug Research, and National Drug Innovative
Program (No.2009ZX09301-011). Support from Priority
Academic Program Development of Jiangsu Higher Education
Institutes (PAPD) is also appreciated.
Supplementary Material
Description of 1H NMR, 13C NMR, HRMS and melting point
of the target compounds. Description of 5-HT1A, 5-HT2A, D1,
D2 and D3 binding assays, [35S]-GTPγS assays and antitumor
assays. Description of molecular modeling. This information is
available via the Internet.
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