Journal of Medicinal Chemistry p. 342 - 358 (2019)
Update date:2022-08-17
Topics:
Bollinger, Sean R.
Engers, Darren W.
Panarese, Joseph D.
West, Mary
Engers, Julie L.
Loch, Matthew T.
Rodriguez, Alice L.
Blobaum, Anna L.
Jones, Carrie K.
Thompson Gray, Analisa
Conn, P. Jeffrey
Lindsley, Craig W.
Niswender, Colleen M.
Hopkins, Corey R.
This work describes the discovery and characterization of novel 6-(1H-pyrazolo[4,3-b]pyridin-3-yl)amino-benzo[d]isothiazole-3-carboxamides as mGlu4 PAMs. This scaffold provides improved metabolic clearance and CYP1A2 profiles compared to previo
View MoreYicheng Goto Pharmaceuticals Co.,Ltd.
Contact:+86 710 3423122
Address:5th Floor,East Gate of Building #2,Servo-Industrial Park,1st Qilin Road,Xiangyang,Hubei,China
Tianjin Boron PharmaTech Co.,Ltd.
Contact:86-022-59845187
Address:B9-401, Tianda Science Park,No.80,4th Avenue,TEDA,Tianjin, China
Lianyungang Ningkang Chemical Co., Ltd
Contact:.+86-518-88588008
Address:http://www.chemnk.com
Nanjing Qirui Material Co., Ltd.
Contact:+86-25-52320053
Address:F4-5, #17 Building, Chuang Yi Yuan, No.6 Guanghua East Street, Nanjing, 210007 P.R.China
Shijiazhuang Haotian Chemical Co., Ltd.
Contact:86-311-85044374
Address:293 Donggang Road
Doi:10.1021/jo01044a002
(1963)Doi:10.1016/j.poly.2008.03.007
(2008)Doi:10.1023/B:CONC.0000018115.15793.d5
(2003)Doi:10.1039/c3nj01293j
(2014)Doi:10.1039/c2ra23043g
(2013)Doi:10.1016/j.electacta.2017.01.071
(2017)