Nucleosides, nucleotides and nucleic acids p. 838 - 852 (2020)
Update date:2022-08-11
Topics:
Takagi-Sato, Miho
Morita, Koji
Onishi, Yoshiyuki
Watahiki, Yuuka
Ishigaki, Taku
Akita, Tomoka
Tomita, Erisa
Kawakami, Junji
Koizumi, Makoto
Oligonucleotides containing 2′-O,4′-C-ethylene nucleic acids (ENA) have been proven highly effective for antisense therapeutics. 2′-O,4′-C-Ethyleneguanosine and its phosphoramidite were previously obtained from 3,5-di-O-benzy1-4-C-(p-tolulenesulfonyloxyet
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