Bioorganic and Medicinal Chemistry Letters p. 1972 - 1977 (2017)
Update date:2022-08-16
Topics:
Xin, Minhang
Hei, Yuan-Yuan
Zhang, Hao
Shen, Ying
Zhang, San-Qi
In this study, a series of new 6-aryl substituted 4-anilinequinazolines was designed and synthesized as PI3Kδ inhibitors based on our reported chemical structures. The preliminary structure-activity relationship (SAR) was established, and compounds 13h an
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