Bioorganic and medicinal chemistry letters (2020)
Update date:2022-08-17
Topics:
Guo, Shanchun
He, Ling
Luo, Lan
Wang, Guangdi
Zhang, Changde
Zhang, Qiang
Zheng, Shilong
Zhong, Qiu
PI-103 (7) is a potent dual phosphatidylinositol 3-kinase (PI3K)/mTOR inhibitor, but its rapid in vivo metabolism hinders its further clinical development. To improve the bioavailability of PI-103, we designed and synthesized a PI-103 bioisostere, PI-103B
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