Archiv der Pharmazie p. 149 - 155 (1995)
Update date:2022-08-30
Topics:
Gorlitzer
Moormann
Pollow
Schaffrath
Starting from the Mannich salt 1 of the aldosterone antagonist canrenone or from 2-methylene-canrenone (2) the A-ring annulated hetero- and carbocycles 5, 6, 8-13 were prepared. Receptor (estradiol, progesterone, androgen, gluco- and mineralocorticoid) binding studies and competition studies with the serum proteins SHBG and CBG were carried out using the compounds 2, 3, 4b, 5, 6b, 8 and 12. The relative binding affinities with CBG are below 1%, in all other cases lower than 0.01%.
View MoreSICHUAN ZHONGBANG NEW MATERIAL CO., LTD
website:http://www.zhongbangst.com
Contact:86-830-2585019
Address:sichuan,china
Shanghai KFSL Pharmaceutical Technology Co.,Ltd.
Contact:+86-21-39971718
Address:859 jiadingchengliu shanghai
HANGZHOU YUNUO CHEMICAL CO.,LTD
website:http://www.yunuochem.com
Contact:0571-83715115
Address:hangzhou
zhengzhou Triz Pharma-Tech Co., Ltd
website:http://www.Trizpharma-tech.com
Contact:+86-0371-86597269,53392065
Address:High-tech Industrial Development Zone, Zhengzhou City, NO.7 Holly Street
Contact:0510-85393305
Address:1619 Huishan Avenue, Huishan District, Wuxi,
Doi:10.1016/j.jallcom.2009.07.163
(2009)Doi:10.1016/0022-328X(89)87090-1
(1989)Doi:10.4067/S0717-97072013000100013
(2013)Doi:10.1002/cssc.202000485
(2020)Doi:10.1006/jcat.2001.3485
(2002)Doi:10.1111/j.1151-2916.2003.tb03361.x
(2003)