tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde

Base Information

• Chemical Name: tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde
• CAS No.: 327605-04-9
• Molecular Formula: C₉H₁₅NO₃
• Molecular Weight: 185.223
• Mol file: 327605-04-9.mol

Synonyms:tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde

Chemical Property of tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde

Chemical Property:

Purity/Quality:

Safty Information:

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MSDS Files:

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Technology Process of tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde

There total 1 articles about tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

carbon monoxide (201230-82-2) + tert-butyl azete-1(2H)-carboxylate (1248510-38-4) → tert-butyl 3-formylazetidine-1-carboxylate (177947-96-5) + tert-butoxycarbonyl-L-azetidine-2-carboxaldehyde (200184-45-8) + tert-butoxycarbonyl-D-azetidine-2-carboxaldehyde (327605-04-9)

Guidance literature:

With 2,2',2'',2'''-(1,2-phenylenebis((1S,3S)-tetrahydro-5,8-dioxo-1H-(1,2,4)diazaphospholo(1,2-a)pyridazine-2,1,3(3H)-triyl))tetrakis(N-(1S)-1-phenylethyl)-benzamide; acetylacetonatodicarbonylrhodium(l); hydrogen; In tetrahydrofuran; toluene; at 35 ℃; for 12h; under 8000.32 Torr; enantioselective reaction;

DOI:10.1021/ja106674n

upstream raw materials:

carbon monoxide

tert-butyl azete-1(2H)-carboxylate

Refernces