103241-34-5Relevant articles and documents
Cholecystokinin Antagonists. Synthesis of Asperlicin Analogues with Improved Potency and Water Solubility
Bock, Mark G.,DiPardo, Robert M.,Rittle, Kenneth E.,Evans, Ben E.,Freidinger, Roger M.,et al.
, p. 1941 - 1945 (2007/10/02)
Seventeen analogues of the selective, competitive cholecystokinin (CCK) antagonist asperlicin 1 were prepared.These compounds were tested as inhibitors of the binding of CCK to rat pancreas and guinea pig brain receptors.Compounds 4, 7, and 8 were m