1046809-84-0

Basic information

• Product Name: (R)-4-[(4-benzyloxy-phenyl)-(4-fluoro-phenylamino)-methyl]-5-oxo-5-((S)-2-oxo-4-phenyl-oxazolidin-3-yl)pentanoic acid benzyl ester
• Synonyms: (R)-4-[(4-benzyloxy-phenyl)-(4-fluoro-phenylamino)-methyl]-5-oxo-5-((S)-2-oxo-4-phenyl-oxazolidin-3-yl)pentanoic acid benzyl ester
• CAS NO: 1046809-84-0
• Molecular Weight: 672.753
• Mol File: 1046809-84-0.mol
• Article Data: 1

Chemical Properties

• CAS DataBase Reference: (R)-4-[(4-benzyloxy-phenyl)-(4-fluoro-phenylamino)-methyl]-5-oxo-5-((S)-2-oxo-4-phenyl-oxazolidin-3-yl)pentanoic acid benzyl ester(CAS DataBase Reference)
• NIST Chemistry Reference: (R)-4-[(4-benzyloxy-phenyl)-(4-fluoro-phenylamino)-methyl]-5-oxo-5-((S)-2-oxo-4-phenyl-oxazolidin-3-yl)pentanoic acid benzyl ester(1046809-84-0)
• EPA Substance Registry System: (R)-4-[(4-benzyloxy-phenyl)-(4-fluoro-phenylamino)-methyl]-5-oxo-5-((S)-2-oxo-4-phenyl-oxazolidin-3-yl)pentanoic acid benzyl ester(1046809-84-0)

Safety Data

• Hazardous Substances Data: 1046809-84-0(Hazardous Substances Data)

Upstream product

• 1046809-83-9 5-oxo-5-((S)-2-oxo-4-phenyl-oxazolidin-3-yl)-pentanoic acid benzyl ester 
• 70627-52-0 4-benzyloxybenzylidene-N-(4-fluoro)phenylanisidine 

Downstream Products

• 1046809-85-1 3-[(2S,3R)-2-(4-benzyloxy-phenyl)-1-(4-fluorophenyl)-4-oxo-azetidin-3-yl]-propionic acid benzyl ester 

Relevant articles and documents

PROCESS FOR PREPARING HIGHLY PURE EZETIMIBE USING NOVEL INTERMEDIATES

The present invention relates to an industrially advantageous process for the preparation of ezetimibe of formula (I) in high yields by using novel benzyl ester intermediates. The present invention further provides a process for the purification of ezetimibe of formula (I).