1104015-93-1Relevant articles and documents
Development of a Practical and Efficient Synthesis of CP-945, 598-01, a CBi Antagonist for the Treatment of Obesity
Ragan, John A.,Bourassa, Dennis E.,Blunt, Jon,Breen, Darragh,Busch, Frank R.,Cordi, Eric M.,Damon, David B.,Do, Nga,Engtrakul, Alanya,Lynch, Denis,McDermott, Ruth E.,Mongillo, Joseph A.,O'Sullivan, Maria M.,Vanderplas, Peter R. RoseBrian C.
experimental part, p. 186 - 197 (2010/04/22)
Development of an efficient bond-forming sequence and optimization of reaction conditions are described for the synthesis of CP-945, 598-01 (1-HC1), a CB, antagonist in clinical studies for the treatment of obesity. Reordering of the bond-forming sequence
