114780-17-5Relevant articles and documents
Stereoselective synthesis and biological activities of O-(E)-1-{1-[6- chloropyridin-3-yhmethyl]-5-methyl-1 H-1,2,3-triazol-4-yl}ethyleneamino-O-ethyl- O-arylphosphorothioates
Zhu, XiaoFei,Chen, XiaoBao,Yan, Man,Shi, De-Qing,Ding, Ke-Rong
, p. 15 - 20 (2008)
To find novel lead compounds having high insecticidal activity, a series of phosphorothioate derivatives containing 1,2,3-triazole and pyridine rings were synthesized by the reaction of 1-{1-[(6-chloropyridin-3-yl)methyl]-5-methyl-1H- 1,2,3-triazol-4-yl}e
Carcarinic acid-1, 2, 3- based triazole compound as well as preparation method and application thereof (by machine translation)
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Paragraph 0217-0219, (2019/12/25)
The method comprises the following steps: firstly 1, 2, 3 - oxidizing and opening the carbon- carbon double bond of the, carcarinic acid into methylene to, obtain carcarinic acid (not shown, in the technical field of, organic 3 - synthesis), Wolf - Kishner - 1, 2, 3 - 1, 2, 3 - 1, 2, 3 - 3 . (by machine translation)
Synthesis and biological activities of O-(E)-(arylmethyl) 1-[1-(arylmethyl)-5-methyl-1H-1,2,3-triazol-4-yl] ethanone oxime ethers
Zhu, Xiao-Fei,Shi, De-Qing
body text, p. 1218 - 1221 (2010/03/04)
(Chemical Equation Presented) A series of novel O-(E)-(arylmethyl) 1-[1-(arylmethyl)-5-methyl-1H-1,2,3-triazol-4-yl] ethanone oxime ethers were synthesized by the O-alkylation of 1-[1-(arylmethyl)-5-methyl-1H-1,2,3-triazol- 4-yl] ethanone oximes with various arylmethyl chlorides in the basic condition. Their structures were confirmed by IR, 1H NMR, mass spectroscopy, and elemental analyses. The preliminary bioassay indicated that some of the target compounds (4a-f) displayed good insecticidal and moderate fungicidal activity. For example, compounds 4c and 4g showed 100% and 90.6% death rates against aphides at the concentration of 250 mg/L, respectively, and compounds 4f and 4g displayed 67% and 78.4% inhibitory rates against Rhizoctonia solani at the dosage of 100 mg/L, respectively.
