1172612-10-0Relevant articles and documents
Design and synthesis of enediyne-peptide conjugates and their inhibiting activity against chymotrypsin
Dutta, Sansa,Basak, Amit,Dasgupta, Swagata
experimental part, p. 3900 - 3908 (2009/10/02)
Novel enediyne-amino acid conjugates 1-4 have been synthesized. All of these effectively target the enzyme chymotrypsin inhibiting its proteolytic activity. The conjugate with a directly linked phenyl alanine is the most effective inhibitor with a Ki