1173981-05-9Relevant articles and documents
Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists
Kojima, Takuto,Mochizuki, Michiyo,Takai, Takafumi,Hoashi, Yasutaka,Morimoto, Sachie,Seto, Masaki,Nakamura, Minoru,Kobayashi, Katsumi,Sako, Yuu,Tanaka, Maiko,Kanzaki, Naoyuki,Kosugi, Yohei,Yano, Takahiko,Aso, Kazuyoshi
, p. 2229 - 2250 (2018/02/21)
A new class of corticotropin releasing factor 1 (CRF1) receptor antagonists characterized by a tricyclic core ring was designed and synthesized. Novel tricyclic derivatives 2a–e were designed as CRF1 receptor antagonists based on con