1224256-32-9Relevant articles and documents
Novel N 2-Substituted pyrazolo[3,4- d ]pyrimidine adenosine A3 receptor antagonists: Inhibition of A3-Mediated human glioblastoma cell proliferation
Taliani, Sabrina,La Motta, Concettina,Mugnaini, Laura,Simorini, Francesca,Salerno, Silvia,Marini, Anna Maria,Da Settimo, Federico,Cosconati, Sandro,Cosimelli, Barbara,Greco, Giovanni,Limongelli, Vittorio,Marinelli, Luciana,Novellino, Ettore,Ciampi, Osele,Daniele, Simona,Trincavelli, Maria Letizia,Martini, Claudia
supporting information; experimental part, p. 3954 - 3963 (2010/08/20)
Adenosine induces glioma cell proliferation by means of an antiapoptotic effect, which is blocked by cotreatment with selective A3 AR antagonists. In this study, a novel series of N2-substituted pyrazolo[3,4-d]pyrimidines 2a-u was de