125112-33-6Relevant articles and documents
HIGHLY FUNCTIONALIZED AZIRIDINES II: A FACILE SYNTHESIS OF DIETHYL AZIRIDINYLPHOSPHONATES AND 2-CHLOROAZIRIDINYLPHOSPHONATES
Coutrot, Philippe,Elgadi, Abdelaziz,Grison, Claude
, p. 1179 - 1192 (1989)
The reaction of diethyl 1-lithio-1-chloromethylphosphonate with aromatic imines gave aziridinylphosphonates in good yields and with an high stereoselectivity.The resulting aziridines reacted with n-BuLi and led to the 2-lithiated anions which were trapped with carbon tetrachloride to give 2-chloroaziridinylphosphonates in excellent yields.