126026-95-7Relevant articles and documents
3-AMINO-2H-AZIRINES IN THE SYNTHESIS OF PEPTIDES: TETRAPEPTIDES WITH α,α-DISUBSTITUTED α-AMINO ACIDS
Sahebi, Mostafa,Wipf, Peter,Heimgartner, Heinz
, p. 2999 - 3010 (2007/10/02)
3-Amino-2,2-dialkyl-2H-azirines 1 are synthons for α,α-disubstituted α-amino acids.Tetrapeptides 15, containing two such amino acids, were synthesized in high yield by application of the "azirine/oxazolone-method".In this versatile approach for the incorp