1270930-62-5Relevant articles and documents
The identification of substituted benzothiophene derivatives as PGE 2 subtype 4 receptor antagonists: From acid to non-acid
Li, Lianhai,Mathieu, Marie-Claude,Denis, Danielle,Therien, Alex G.,Wang, Zhaoyin
scheme or table, p. 734 - 737 (2011/03/18)
We disclose herein our preliminary SAR study on the identification of substituted benzothiophene derivatives as PGE2 subtype 4 receptor antagonists. A potent EP4 antagonist 6a (Ki = 1.4 nM with 10% HSA) was identified. Fur