128832-34-8Relevant articles and documents
Novel Acyl-CoA:Cholesterol Acyltransferase Inhibitors. Synthesis and Biological Activity of 3-Quinolylurea Derivatives
Tawada, Hiroyuki,Harcourt, Myles,Kawamura, Noriaki,Kajino, Masahiro,Ishikawa, Eiichiro,et al.
, p. 2079 - 2084 (2007/10/02)
A series of 3-quinolylurea derivatives (1) was synthesized and evaluated for acyl-CoA:cholesterol acyltransferase (ACAT) inhibitory activity.For in vitro studies, the most potent inhibitory activity was found in derivatives having substituents at the 6,7-