1304685-27-5Relevant articles and documents
Copper-catalyzed electrophilic amination of heteroaromatic and aromatic C-H bonds via TMPZnCl.·LiCl mediated metalation
McDonald, Stacey L.,Hendrick, Charles E.,Bitting, Katie J.,Wang, Qiu
, p. 356 - 372 (2016/08/23)
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Copper-catalyzed direct amination of polyfluoroarenes and azoles with hydroxylamines and its application to the synthesis of 3-aminobenzoheteroles
Matsuda, Naoki,Hirano, Koji,Satoh, Tetsuya,Miura, Masahiro
experimental part, p. 1792 - 1797 (2012/07/28)
A copper-catalyzed electrophilic, umpolung amination strategy for the direct C-H amination of polyfluoroarenes and 1,3-azoles has been developed. The copper-based amination reaction is robust and can be easily scaled up on a gram scale. Its application to