13423-60-4Relevant articles and documents
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Grundmann,Raetz
, p. 1037 (1956)
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Deprotometalation-iodolysis and computed CH acidity of 1,2,3- and 1,2,4-triazoles. Application to the synthesis of resveratrol analogues
Nagaradja, Elisabeth,Bentabed-Ababsa, Ghenia,Scalabrini, Mathieu,Chevallier, Floris,Philippot, Stéphanie,Fontanay, Stéphane,Duval, Rapha?l E.,Halauko, Yury S.,Ivashkevich, Oleg A.,Matulis, Vadim E.,Roisnel, Thierry,Mongin, Florence
, p. 6355 - 6363 (2015)
1-Aryl- and 2-aryl-1,2,3-triazoles were synthesized by N-arylation of the corresponding azoles using aryl iodides. The deprotometalations of 1-phenyl-1,2,3-triazole and -1,2,4-triazole were performed using a 2,2,6,6-tetramethylpiperidino-based mixed lithi
A ligand-free copper-catalyzed strategy to the N-arylation of indazole using aryl bromides
Bai, Di-Xiang,Lim, Rachel Sin-Ee,Ng, Hui-Fen,Teo, Yong-Chua
supporting information, p. 1398 - 1405 (2021/03/08)
A simple and efficient strategy for the C–N cross-coupling of indazole with a variety of substituted aryl bromides is reported. Under the optimized conditions, a broad scope of N-arylated products were obtained in good to excellent yields (up to 87%) under the ligand-free conditions.
Facile One-Pot Synthesis of Methyl 1-Aryl-1H-1,2,4-triazole-3-carboxylates from Nitrilimines with Vilsmeier Reagent
Tsai, Shuo-En,Chiang, Kun-Heng,Tseng, Ching-Chun,Chen, Nai-Wei,Chern, Ching-Yuh,Wong, Fung Fuh
, p. 1754 - 1762 (2019/02/24)
Two convenient and effective one-pot methods have been developed to synthesize methyl 1-aryl-1H-1,2,4-triazole1–3-carboxylates by using hydrazonoyl hydrochlorides (nitrilimines) with Vilsmeier reagent. The first, a direct one-pot method, involved the reac