1349179-60-7Relevant articles and documents
Identification of a novel RAMP-independent CGRP receptor antagonist
Zartman, C. Blair,Bell, Ian M.,Gallicchio, Steven N.,Graham, Samuel L.,Kane, Stefanie A.,Mallee, John J.,Rutledge, Ruth Z.,Salvatore, Christopher A.,Vacca, Joseph P.,Williams, Theresa M.
, p. 6705 - 6708 (2011)
Identification of an HIV integrase inhibitor with micromolar affinity for the CGRP receptor led to the discovery of a series of structurally novel CGRP receptor antagonists. Optimization of this series produced compound 16, a low-molecular weight CGRP rec
