1350522-74-5Relevant articles and documents
Design, synthesis and biological activity of original pyrazolo-pyrido- diazepine, -pyrazine and -oxazine dione derivatives as novel dual Nox4/Nox1 inhibitors
Gaggini, Francesca,Laleu, Beno?t,Orchard, Mike,Fioraso-Cartier, Laetitia,Cagnon, Laurne,Houngninou-Molango, Sophie,Gradia, Angelo,Duboux, Guillaume,Merlot, Cédric,Heitz, Freddy,Szyndralewiez, Cédric,Page, Patrick
, p. 6989 - 6999 (2012/01/03)
Pyrazolo-pyrido-diazepine, -pyrazine and -oxazine dione derivatives are new chemical entities with good and attractive druglikeness properties. A series of pyrazolo-pyrido-diazepine dione analogs demonstrated to be particularly amenable to lead optimizati